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Optimization of Azaspirooxindolinone-based PROTACs targeting BTK: Synthesis, kinase profiling, and degradation analysis

RAMPEESA, N., R. GUNDLA, S. GURSKÁ, S. YADAM, S. TANGALLAPALLI, S. ANUGU, J. DE SANCTIS, P. DŽUBÁK, M. HAJDÚCH, N. KATARI, V. DAS, S. JONNALAGADDA
Optimization of Azaspirooxindolinone-based PROTACs targeting BTK: Synthesis, kinase profiling, and degradation analysis. Results in Chemistry. 2026, 23, 103145, ISSN: 2211-7156,  PDF.